Both AP-7 and D-AP7 function as potent, specific antagonists of the NMDA receptor.
2.
The discovery of EPAC specific antagonists represents a research milestone that allows the pharmacological manipulation of EPAC activity.
3.
SIADH can also be treated with specific antagonists of the ADH receptors, such as conivaptan or tolvaptan.
4.
Scientists proposed that specific antagonists can act on GABAergic interneurons, enhancing cortical inhibition and preventing excessive glutamatergic transmission associated with schizophrenia.
5.
Application of CB 2-specific antagonists has found that these receptors are also involved in mediating analgesic effects in the peripheral nervous system.
6.
Nelivaptan ( SSR149415 ) and D-[ Leu 4-Lys 8 ]-vasopressin are a specific antagonist and agonist for the vasopressin 1b receptor, respectively.
7.
The other specific antagonist you may hear about is flumazenil, which antagonises a benzodiazepine coma ( for which naloxone won't work ) .-- Seejyb 15 : 39, 15 December 2006 ( UTC)
8.
LY-404, 039 possesses partial agonist actions at D 2 receptors and inhibits the binding of the D 2-specific antagonist HVA in the prefrontal cortex in a manner similar to the atypical antipsychotic clozapine.
9.
While only those who belong to Bowser or specific antagonists are enemies to Mario or players, other members of these species ( usually individuals ) have their own life in or out of Mushroom Kingdom ( e . g.
10.
ICI-118, 551 has no known therapeutic use in humans although it has been used widely in research to understand the action of the ? 2 adrenergic receptor, as few other specific antagonists for this receptor are known.